AAIPHARMA
SERVICES SEARCH:
ProLiquitab
Bioavailability Enhancement
Self Emulsified System in a Tablet
Solubilized Drug Emulsion Adsorbed onto Solid Carrier
Proprietary combinations of Excipients for Enhanced Solubility
Manufacturing Process
1. Disperse/Dissolve API into SEDDS
2. Adsorb SEDDS onto Solid Carrier
3. Granulate API Loaded Carrier
4. Blend with Additional Excipients
5. Tablet Compression
Graphic Depiction of ProLiquitab Matrix
ProLiquitab Comparison with Capsule Dosage Form
Potential Benefits:
Improved Therapy
More rapid onset vs conventional tablet
Improved bioavailability
Lower PK variability
Higher blood levels
Lower API requirements
Patient Preferred Tablet Dosage Form
Solutions for poorly absorbable compounds:
Solutions for poorly soluble compounds:
Controlled and prolonged release profiles:
Site specific delivery in the GI tract:
Life cycle management and line extensions:
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